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Innovative tools for breast cancer research and drug discovery

Breast cancer is the most common cancer in women worldwide. It is highly heterogeneous with distinct breast cancer types and subtypes, posing challenges for diagnosis and treatment. There are four key molecular breast cancer subtypes classified based on the expression of oestrogen and progesterone hormone receptors (ER and PR) and human epidermal growth factor receptor 2 (HER2). These include luminal A, luminal B, HER2-positive, and triple-negative breast cancer (TNBC), which is characterised by the lack of expression of any of the above receptors. TNBC is the most challenging breast cancer type as it does not respond to any hormonal or HER2-targeted therapies.

There is a need for breast cancer models that capture its heterogeneity to uncover novel disease mechanisms underlying its complexity and for more precise drug development.

At CancerTools.org, we have curated an extensive collection of breast cancer research tools, deposited by scientists from academic universities and leading cancer centres over 40 years. This includes a diverse array of breast cancer cell lines for improved disease modelling, more complex in vivo patient derived xenograft (PDX) and mouse models to enhance preclinical drug discovery workflows, as well as widely used antibodies to study tumour signalling pathways.

Explore our breast cancer research tools collection

Disease modelling

CancerTools provides diverse breast cancer cell lines to accurately model the tumour-microenvironment, metastases, and treatment resistance, to aid scientists uncover new pathways and develop improved in vitro models of breast cancer.

MCF-7/S0.5 cells stained for oestrogen receptor expression

Anti-oestrogen resistant MCF7 and T47D cell lines

These have been derived from human breast cancer cell lines, MCF7 and T47D which depend on oestrogen for growth and demonstrate resistance to hormone-dependent breast cancer treatments. These anti-oestrogen resistant lines, including the MCF7/TAMR-1 cell line, allow researchers to better understand the underlying molecular mechanisms of resistance.

MCF-7/S0.5 cells stained for oestrogen receptor expression
MCF10A-HER2 cells cultured in 3D formed flat projecting cells of complex masses, typical of transformed cells. Adapted from Hayat A. et al. 2023. Dis Model Mech. Feb 1;16(2). PMID: 36661191.

HER2-positive MCF10A derivative line

This MCF10A breast cancer subline shows inducible overexpression of the HER2 protein at clinically relevant levels, co-expresses GFP for tracking and selection, and can be cultured in 3D for enhanced biological relevance. This cell line enables early molecular change detection in HER2-driven tumour development and HER2-mediated signalling pathway analysis.

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Breast cancer cells resisting treatment. Contributed by Saumya Samadhiya

Triple negative MDA-MB-231 modified reporter line

The MDA-MB-231/ EGFP_LC3 cell line is a triple negative breast cancer (TNBC) subtype line that stably expresses the EGFP tagged microtubule associated protein 1 light chain 3 beta (MAP1LC3B) protein, a key player in the autophagy pathway. These cells can be used to study autophagy pathway dynamics in real-time and study autophagy-mediated therapy resistance, in TNBC.

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Breast cancer cells resisting treatment. Contributed by Saumya Samadhiya

Gene-edited MCF7 and MDA-MB-231 cell lines

Gene-edited MCF7 sgRNA 1 & 2 and MDA-MB-231 sgRNA 1 & 2 cell lines enable the investigation of the breast BRCA1 non mutated and hypermethylated breast cancer tumourigenesis pathways. Both cell lines contain site-specific methylations in the BRCA1 promoter.

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Plasmax™: a physiologically relevant cell culture medium

Plasmax is a defined cell culture medium that provides a physiologically relevant environment by mirroring the concentration of over 50 components found in human plasma. This media been used to successfully culture three triple-negative breast cancer cell lines, BT549, MDA-MB-468 and CAL-120, by recapitulating the tumour metabolic environment.

Explore our breast cancer cell lines

Tool nameCat. #Inventor/ InstituteOrganismKey attributes
MCF7/S0.5   152090 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen/fulvestrant sensitive control line 
MCF7/TAMR-1  152089 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen resistant subline 
MCF7/TAMR-4152088 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen resistant subline
MCF7/TAMR-7  152087Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen resistant subline 
MCF7/TAMR-8152086 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen resistant subline 
MCF7/164R-1152091 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
MCF7/164R-4 152101 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
MCF7/164R-5  152102 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
MCF7/164R-7  152103 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
MCF7/182R-1152104 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
MCF7/182R-6  152105 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
MCF7/182R-7 152106 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
T47D/S2 152109 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen sensitive control line 
T47D/TR-1  152108 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen resistant subline 
T47D/TR-2  152110 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Tamoxifen resistant subline 
T47D/S5152111Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant sensitive control line 
T47D-182R2 151890 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
T47D-182R1 151891 Anne Lykkesfeldt, 
Danish Cancer Society 
Human– Fulvestrant resistant subline 
MCF10A-HER2 157986 Richard Grose, Gabriella Ficz and Ateequllah Hayat, 
Queen Mary University of London 
Human– Inducible HER2 overexpression at clinically relevant levels 
– Integrated GFP expression 
SK-BR-3161911 Lloyd J. Old and Germain 
Trempe, Memorial Sloan -Kettering Cancer Center 
(MSK) 
Human– Human cell line 
– Overexpresses HER2 protein 
MDA-MB-231/ EGFP_LC3161138 T. R. Santhosh Kumar,
Rajiv Gandhi Centre for Biotechnology
Human– TNBC line stably expressing  EGFP tagged LC3 protein 
– Recapitulates LC3 puncta
formation 
E3 STn 151847 Joyce Taylor-Papadimitriou 
and Joy Burchell,
Cancer Research UK, London Research Institute 
Mouse– Mouse cell line 
– Expresses human MUC1
and Sialyl-Tn 

Drug discovery

CancerTools.org provides anti-oestrogen resistant cell lines, patient-derived organoid (PDO) and patient-derived xenograft (PDXs) breast cancer models that capture tumour heterogeneity and are clinically relevant, to enhance breast cancer drug discovery.

MCF-7/S0.5 cells stained for oestrogen receptor expression

Anti-oestrogen resistant MCF7 and T47D cell lines

These anti-oestrogen resistant cell lines, as described earlier, offer the potential for developing novel predictive biomarkers for therapy response and an improved understanding of the underlying molecular mechanisms of resistance, supporting new drug discovery.

MCF-7/S0.5 cells stained for oestrogen receptor expression

Patient-derived xenograft (PDX) models

PDX models are created by transplanting human tumour tissue into immunodeficient mice. Our collection of breast cancer PDX models includes those from patients affected by the most advanced and lethal forms of breast cancer, such as aggressive, metastatic and treatment resistant subtypes. PDX models are superior in recapitulating patient tumour characteristics including spatial structure, intratumour heterogeneity, genomic features, tumour growth rates, metastatic patterns and drug responses. These highly translatable models can be used to enhance and de-risk preclinical in vivo drug validation.

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Explore our breast cancer PDX models

Tool nameCat. #Inventor/ InstituteKey attributes
HCI-001 to HCI-054 breast cancer PDX 162069 to 162121 Alana L. Welm, Yi-Chun Lin and Yoko Sakata DeRose, 
The University of Utah Research Foundation 
– Capture patient 
intratumour heterogeneity 
– Recapitulate patient drug
response profiles 
Mouse icon

MUC1 mouse model

Tumour associated antigen, MUC1 is aberrantly overexpressed in 90% of human breast cancers and represents a promising therapeutic target for breast cancer. Our MUC1 mouse model can be used for the preclinical study of anti-MUC1 vaccines/immunotherapies.

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Mouse icon

Tumour signalling

CancerTools.org provides widely used antibodies for targets with key functions in tumour signalling pathways including tumour suppressors (p53, RB1), oncogenes (c-MYC), and tumour associated antigens (MUC1).

Tumour suppressors

Antibodies targeting p53, Retinoblastoma 1 (RB1), and Maspin, all tumour suppressors with key roles in biological processes across different types of tumours including breast cancer tumours. Our collection also features antibodies against PALB2 and BRCA1/2, both tumour suppressors whose pathogenic variants are associated with breast cancer, as well as ovarian and pancreatic cancers.

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Oncogenes

Multiple antibodies targeting the oncogene, c-MYC, a transcription factor of high interest in breast cancer research due to its regulation of key biological processes in the tumour microenvironment, e.g. angiogenesis, tumour evasion, invasion, and migration

Access oncogenes

Tumour associated antigens

Antibodies targeting tumour associated antigens like MUC1, a promising marker for breast cancer diagnosis and prognosis.

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Explore our breast cancer antibodies

Tool nameCat. #Inventor/ InstituteReactivityKey attributes
Anti-cMyc [9E10] 151067 Gerard Evan,
University of California San Francisco 
Human– Monoclonal antibody 
– Detects c-Myc oncogene product 
Anti-MUC1 [HMFG1] 151495 Joyce Taylor-Papadimitriou 
and Joy Burchell,
Cancer Research UK, London 
Research Institute 
Human– Monoclonal antibody 
– Detects human MUC-1 

Tool enquiry

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