MZ1 small molecule (tool compound)

(+)-JQ1 based PROTAC that selectively degrades BRD4 in cells

Contributors

Inventor Institute
Alessio Ciulli ; Michael Zengerle ; Kwok-Ho Chan University of Dundee
Cat. #: 158364
Research Fields: Genetics
Alternate name: BRD4, CAP, bromodomain containing 4, chromosome-associated protein, HUNK1, HUNKI, MCAP
Product description: (+)-JQ1 based PROTAC that selectively degrades BRD4 in cells
Molecular weight: 1002.64
Primary target: BRD4
Shipping conditions: Dry Ice
Solubility: DMSO; Ethanol
References:

Zengerle et al. 2015. ACS Chem Biol. 10(8):1770-7. PMID: 26035625.

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