#153191

CDK inhibitor BS-194 Small Molecule (Tool Compound)

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Cat. #153191

CDK inhibitor BS-194 Small Molecule (Tool Compound)

Cat. #: 153191

Sub-type: Inhibitor

Availability: Please enquire for quantities and pricing

This fee is applicable only for non-profit organisations. If you are a for-profit organisation or a researcher working on commercially-sponsored academic research, you will need to contact our licensing team for a commercial use license.

Contributor

Inventor: Simak Ali

Institute: Imperial College London

Tool Details
Handling
Target Details
Related Tools
References

Tool Details

*FOR RESEARCH USE ONLY

  • Tool name: CDK inhibitor BS-194 Small Molecule (Tool Compound)
  • Research fields: Cancer;Genetics
  • Molecular formula: C20H27N5O3
  • Tool sub type: Inhibitor
  • Description: BS-194 is a selective and potent CDK inhibitor, which inhibits CDK2, CDK1, CDK5, CDK7, and CDK9.
  • Purpose: Inhibitor
  • Selectivity: CDK1, CDK2, CDK7, and CDK9
  • Iupac: (2S,3S)-3-(7-(benzylamino)-3- isopropylpyrazolo[1,5-a]pyrimidin-5- ylamino)butane-1,2,4-triol
  • Molecular weight: 385.5

Handling

  • Purity: 385.5 g/mol
  • Storage conditions: Ambient
  • Shipping conditions: Dry Ice

Target Details

  • Ic50: CDK2, CDK1, CDK5, CDK7, and CDK9 (IC50=3, 30, 30, 250, and 90 nmol/L, respectively)

Related Tools

  • Related tools: CDK7 inhibitor BS-181 Small Molecule (Tool Compound)

References

  • J. Med. Chem. 2010, 53, 8508–8522